VECLADX Venetoclax 100mg

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Key Highlights

Venetoclax, b -2(BCL-2) ,BCL-2 , , BCL-2 BCL-2 , , ,

Service Promise

Direct from JapanLicensed PharmacyPharmacist CheckedEditable in Admin

Specifications

Specification
100mg*112 tablets

Product Info

English Name
Venetoclax 100mg
Chinese Name
VECLADX
Generic Name
VECLADX

Specifications

Specification
100mg*112 tablets

Full Details

Indications

VECLADX , 17p CLL VENTCLEXTA

How It Works

12.1 How It Works BCL-2 ,BCL-2 CLL AML BCL-2 ,BCL-2 , BCL-2 , BIM , caspase , , BCL-2

Pharmacology

12 12.1 How It Works BCL-2 ,BCL-2 BCL-2 CLL AML , , BCL-2 , BIM , caspase , , BCL-2 12.2 - , CLL/SLL AML

Dosage

• VECLADX , VENTCLEXTA VECLADX • VECLADX o VECLADX TLS o VENTCLEXTA 5 , VENTCLEXTA • Description • VECLADX 1 • VECLADX • VECLADX 8 , VECLADX 8 , • VECLADX ,

Precautions

5 Precautions (TLS) TLS , 2.4,5.1 ,

Contraindications

4. / CLL/SLL , VENCLEXTA CYP3A , [ Dosage (2.6) (7.1)] / CLL/SLL , CYP3A (2.6, 4, 7.1)

Drug Interactions

7 CYP3A P-gp (2.6, 7.1) CYP3A (7.1) P-gp 6 (7.2) 7.1 CYP3A P-gp CYP3A P-gp Cmax AUC0-INF [ (12.3)], , (TLS) [ Precautions (5.1)] CLL/SLL , CYP3A [ 4 ]

Adverse Reactions

(TLS) TLS TLS , , VECLADX , TLS VENTCLEXTA , , TLS (IV) 5 , VECLADX TLS VECLADX TLS , , • • • • • • • • • • • VECLADX TLS 6 8 56 , 2 , VECLADX , , VENTCLEXTA • VECLADX , VECLADX , VECLADX , VECLADX o o o o o o VECLADX , , VENTCLEXTA

Storage

• VECLADX 86°F (30°C) • 4 VENTCLEXTA VENTCLEXTA

Package Insert

Ingredients

11 Description BCL-2 , C₄₅H₅₀ClN₇O₇S, 868.44 4-(4-{[2-(4- )-4,4- -1- -1- ] } -1- )-N-({3- -4-[( -2H- -4- ) ] } )-2-(1H- [2,3-b] -5- ) ), VENCLEXTA , 10 mg 50 mg 100 mg venetoclax 80

Indications

VECLADX , 17p CLL VENTCLEXTA

Dosage

• VECLADX , VENTCLEXTA VECLADX • VECLADX o VECLADX TLS o VENTCLEXTA 5 , VENTCLEXTA • Description • VECLADX 1 • VECLADX • VECLADX 8 , VECLADX 8 , • VECLADX ,

Adverse Reactions

(TLS) TLS TLS , , VECLADX , TLS VENTCLEXTA , , TLS (IV) 5 , VECLADX TLS VECLADX TLS , , • • • • • • • • • • • VECLADX TLS 6 8 56 , 2 , VECLADX , , VENTCLEXTA • VECLADX , VECLADX , VECLADX , VECLADX o o o o o o VECLADX , , VENTCLEXTA

Contraindications

4. / CLL/SLL , VENCLEXTA CYP3A , [ Dosage (2.6) (7.1)] / CLL/SLL , CYP3A (2.6, 4, 7.1)

Precautions

5 Precautions (TLS) TLS , 2.4,5.1 ,

Use in Pregnancy and Lactation

8.1 How It Works[ 12.1 ],VENCLEXTA - VENCLEXTA , , , 400 mg/ 1.2 AUC , ,

Drug Interactions

7 CYP3A P-gp (2.6, 7.1) CYP3A (7.1) P-gp 6 (7.2) 7.1 CYP3A P-gp CYP3A P-gp Cmax AUC0-INF [ (12.3)], , (TLS) [ Precautions (5.1)] CLL/SLL , CYP3A [ 4 ]

Overdose

10. VENCLEXTA , , , TLS [ Dosage 2.2 2.3 2.4 2.5 ] ,

Clinical Pharmacology

12 12.1 How It Works BCL-2 ,BCL-2 BCL-2 CLL AML , , BCL-2 , BIM , caspase , , BCL-2 12.2 - , CLL/SLL

Pharmacology and Toxicology

13 13.1 6 Tg.rasH2 , M27 400 mg/kg/ , 250 mg/kg/ M27 Ames , , , 835 mg/kg M27 Ames

Clinical Studies

14 1. AMPLIFY IRC Kaplan-Meier 1 2 3 4 14.1 / AMPLIFY (ACE-CL-311) (NCT03836261), VENCLEXTA (VEN+A) del(17p) TP53 18 CLL VENCLEXTA acalabrutinib VEN+A 1 1 , 100 mg Acalabrutinib, 14 , 3 1 , VENCLEXTA 5 , 20 mg,

Storage

• VECLADX 86°F (30°C) • 4 VENTCLEXTA VENTCLEXTA

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Description

Indications

VECLADX , 17p CLL VENTCLEXTA

How It Works

12.1 How It Works BCL-2 ,BCL-2 CLL AML BCL-2 ,BCL-2 , BCL-2 , BIM , caspase , , BCL-2

Pharmacology

12 12.1 How It Works BCL-2 ,BCL-2 BCL-2 CLL AML , , BCL-2 , BIM , caspase , , BCL-2 12.2 - , CLL/SLL AML

Dosage

• VECLADX , VENTCLEXTA VECLADX • VECLADX o VECLADX TLS o VENTCLEXTA 5 , VENTCLEXTA • Description • VECLADX 1 • VECLADX • VECLADX 8 , VECLADX 8 , • VECLADX ,

Precautions

5 Precautions (TLS) TLS , 2.4,5.1 ,

Contraindications

4. / CLL/SLL , VENCLEXTA CYP3A , [ Dosage (2.6) (7.1)] / CLL/SLL , CYP3A (2.6, 4, 7.1)

Drug Interactions

7 CYP3A P-gp (2.6, 7.1) CYP3A (7.1) P-gp 6 (7.2) 7.1 CYP3A P-gp CYP3A P-gp Cmax AUC0-INF [ (12.3)], , (TLS) [ Precautions (5.1)] CLL/SLL , CYP3A [ 4 ]

Adverse Reactions

(TLS) TLS TLS , , VECLADX , TLS VENTCLEXTA , , TLS (IV) 5 , VECLADX TLS VECLADX TLS , , • • • • • • • • • • • VECLADX TLS 6 8 56 , 2 , VECLADX , , VENTCLEXTA • VECLADX , VECLADX , VECLADX , VECLADX o o o o o o VECLADX , , VENTCLEXTA

Storage

• VECLADX 86°F (30°C) • 4 VENTCLEXTA VENTCLEXTA

Additional information

Specification

100mg*112片