Lucius Sunitinib online kaufen

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Pharmacie physique à Hong Kong, authenticité 100% garantie

Points forts

1.1 (GIST) 1.2 (RCC) 1.3 RCC 1.4

Garanties de service

Expédition transfrontalièrePharmacie agrééeContrôle pharmacienGarantie authenticité

Caractéristiques

Spécification
12.5mg*28 25mg*28 50mg*28
Fabricant
Lucius Pharmaceuticals
Expédition
Hong Kong
SKU : ND Catégorie : Étiquettes : , , Marque :

Informations produit

Nom anglais
Sunitinib
Nom générique
Sunitinib

Caractéristiques

Spécification
12.5mg*28 25mg*28 50mg*28
Fabricant
Lucius Pharmaceuticals
Expédition
Hong Kong

Détails complets

Indications

1.1 (GIST) 1.2 (RCC) 1.3 RCC 1.4

Mécanisme d’action

, RTK , >80 , PDGFRα PDGFRβ VEGFR1 VEGFR2 VEGFR3 KIT Fms -3 FLT3 1 CSF-1R RET

Pharmacologie

12.1 Mecanisme d action , RTK , >80 , PDGFRα PDGFRβ VEGFR1 VEGFR2 VEGFR3 KIT Fms -3 FLT3 1 CSF-1R RET

Posologie

2.1 (GIST) (RCC) (GIST) (RCC) 50 mg, 4 2 4/2 , 2.2 (RCC) (RCC) 50 mg, 4 2 4/2 , 9 6 2.3 (pNET) (pNET) 50 mg, 4 2 4/2 , 9 6

Interactions médicamenteuses

7.1 CYP3A4 CYP3A4 [ (12.3)] CYP3A4 , [ Posologie(2.5)] CYP3A4 CYP3A4 [ (12.3)]

Effets indésirables

Description [ Precautions (5.1)] [ Precautions (5.2)] QT [ Precautions (5.3)] [ Precautions (5.4)] [ Precautions (5.5)] [ Precautions (5.6)] [ Precautions (5.7)] [ Precautions (5.8)] [ Precautions (5.9)] [ Precautions (5.10)] [ Precautions (5.10)]

Package Insert

Indications

1.1 (GIST) 1.2 (RCC) 1.3 RCC 1.4

Posologie

2.1 (GIST) (RCC) (GIST) (RCC) 50 mg, 4 2 4/2 , 2.2 (RCC) (RCC) 50 mg, 4 2 4/2 , 9 6 2.3 (pNET) (pNET) 50 mg, 4 2 4/2 , 9 6

Effets indésirables

Description [ Precautions (5.1)] [ Precautions (5.2)] QT [ Precautions (5.3)] [ Precautions (5.4)] [ Precautions (5.5)] [ Precautions (5.6)] [ Precautions (5.7)] [ Precautions (5.8)] [ Precautions (5.9)] [ Precautions (5.10)] [ Precautions (5.10)]

Use in Pregnancy and Lactation

8.1 Mecanisme d action, [ 12.1 ] , , , RDD 50 mg AUC 5.5 0.3

Interactions médicamenteuses

7.1 CYP3A4 CYP3A4 [ (12.3)] CYP3A4 , [ Posologie(2.5)] CYP3A4 CYP3A4 [ (12.3)]

Clinical Pharmacology

12 12.1 Mecanisme d action , (RTK), >80 , (PDGFRα PDGFRβ) (VEGFR1 VEGFR2 VEGFR3) (KIT) Fms -3 (FLT3) 1 (CSF-1R) (RET) RTK ,

Pharmacology and Toxicology

13 13.1 rasH2 Sprague-Dawley rasH2 , 1 6 , ≥25 mg/kg/ , / , 8 mg/kg/ , rasH2 , , 28 , 7 , 1 mg/kg/ AUC 0.9 ,

Clinical Studies

14 14.1 1 1 (NCT#00075218) , (GIST) (TTP) (PFS) (ORR) (OS) 2:1 , 50 mg , , 4/2,

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Description

Indications

1.1 (GIST) 1.2 (RCC) 1.3 RCC 1.4

Mécanisme d’action

, RTK , >80 , PDGFRα PDGFRβ VEGFR1 VEGFR2 VEGFR3 KIT Fms -3 FLT3 1 CSF-1R RET

Pharmacologie

12.1 Mecanisme d action , RTK , >80 , PDGFRα PDGFRβ VEGFR1 VEGFR2 VEGFR3 KIT Fms -3 FLT3 1 CSF-1R RET

Posologie

2.1 (GIST) (RCC) (GIST) (RCC) 50 mg, 4 2 4/2 , 2.2 (RCC) (RCC) 50 mg, 4 2 4/2 , 9 6 2.3 (pNET) (pNET) 50 mg, 4 2 4/2 , 9 6

Interactions médicamenteuses

7.1 CYP3A4 CYP3A4 [ (12.3)] CYP3A4 , [ Posologie(2.5)] CYP3A4 CYP3A4 [ (12.3)]

Effets indésirables

Description [ Precautions (5.1)] [ Precautions (5.2)] QT [ Precautions (5.3)] [ Precautions (5.4)] [ Precautions (5.5)] [ Precautions (5.6)] [ Precautions (5.7)] [ Precautions (5.8)] [ Precautions (5.9)] [ Precautions (5.10)] [ Precautions (5.10)]

Informations complementaires

Specification

12.5mg*28粒, 25mg*28粒, 50mg*28粒