Description
Indications
1.1 (GIST) 1.2 (RCC) 1.3 RCC 1.4
How It Works
, RTK , >80 , PDGFRα PDGFRβ VEGFR1 VEGFR2 VEGFR3 KIT Fms -3 FLT3 1 CSF-1R RET
Pharmacology
12.1 How It Works , RTK , >80 , PDGFRα PDGFRβ VEGFR1 VEGFR2 VEGFR3 KIT Fms -3 FLT3 1 CSF-1R RET
Dosage
2.1 (GIST) (RCC) (GIST) (RCC) 50 mg, 4 2 4/2 , 2.2 (RCC) (RCC) 50 mg, 4 2 4/2 , 9 6 2.3 (pNET) (pNET) 50 mg, 4 2 4/2 , 9 6
Drug Interactions
7.1 CYP3A4 CYP3A4 [ (12.3)] CYP3A4 , [ Dosage(2.5)] CYP3A4 CYP3A4 [ (12.3)]
Adverse Reactions
Description [ Precautions (5.1)] [ Precautions (5.2)] QT [ Precautions (5.3)] [ Precautions (5.4)] [ Precautions (5.5)] [ Precautions (5.6)] [ Precautions (5.7)] [ Precautions (5.8)] [ Precautions (5.9)] [ Precautions (5.10)] [ Precautions (5.10)]





